Escitalopram (Lexapro)

Class

SSRI (Selective Serotonin Reuptake Inhibitor)

Mechanism

Highly selective serotonin reuptake inhibitor (SERT), enhancing serotonergic neurotransmission.

FDA-Approved Use

Major depressive disorder (MDD), generalized anxiety disorder (GAD)

Off-Label Use

Binge eating disorder, obsessive-compulsive disorder (OCD), posttraumatic stress disorder (PTSD), panic disorder, social anxiety disorder (SoAD), premenstrual dysphoric disorder (PMDD), vasomotor symptoms, fibromyalgia, post-stroke depression (PSD), depression in Parkinson’s disease (PD), depression in dementia

Formulation

Oral tablets (5 mg, 10 mg, 20 mg)

Titration

5–10 mg p.o. daily, titrating as clinically indicated

Dose Range

10–20 mg/day

Kinetics

Half-life ~27–32 hours; metabolized primarily by CYP3A4 and CYP2C19; steady state in ~1 week

Common AEs

Headache, nausea, insomnia, fatigue, dry mouth, somnolence, sexual dysfunction

Serious/Rare AEs

QTc prolongation (especially at higher doses or with other QT-prolonging agents), serotonin syndrome, hyponatremia

Monitoring

Monitor ECG if combined with other QT-prolonging agents or in patients with cardiac risk factors; monitor for serotonin syndrome and suicidality

Black Box Warning

Increased risk of suicidal thoughts and behaviors in children, adolescents, and young adults with MDD and other psychiatric disorders

Considerations

Escitalopram may reduce neuropsychiatric symptoms in post-stroke depression and vascular cognitive impairment. It is preferred in patients with seizure disorders due to fewer CYP450 interactions compared to other SSRIs. Use cautiously in hepatic impairment or patients with electrolyte abnormalities. QTc prolongation risk increases with higher doses or concomitant use of other QT-prolonging medications.