Citalopram (Celexa)

Class

SSRI (Selective Serotonin Reuptake Inhibitor)

Mechanism

Selective serotonin reuptake inhibitor (SERT), increasing serotonergic neurotransmission.

FDA-Approved Use

Major depressive disorder (MDD)

Off-Label Use

Generalized anxiety disorder (GAD), obsessive-compulsive disorder (OCD), panic disorder, post-stroke affective lability, post-stroke depression, depression in Parkinson’s disease (PD), depression in dementia, agitation and aggression in neurodevelopmental disabilities

Formulation

Oral tablets (10 mg, 20 mg, 40 mg)

Titration

10–20 mg p.o. daily, titrating to 20–40 mg/day as tolerated; maximum dose in adults >60 years is 20 mg/day due to QTc prolongation risk

Dose Range

20–40 mg/day (max 20 mg/day in elderly >60 years)

Kinetics

Half-life ~35 hours; metabolized primarily via CYP2C19 and CYP3A4; steady state in ~1 week

Common AEs

Nausea, dry mouth, sexual dysfunction, sedation

Serious/Rare AEs

QTc prolongation, serotonin syndrome, hyponatremia

Monitoring

ECG monitoring recommended for patients with cardiac risk factors or on QT-prolonging medications; monitor electrolytes especially in elderly

Black Box Warning

Increased risk of suicidal thoughts and behaviors in children, adolescents, and young adults with MDD and other psychiatric disorders

Considerations

Citalopram is frequently used to manage behavioral symptoms of dementia, particularly agitation and impulsivity. It requires ECG monitoring in patients with cardiac risk factors, especially those with QT prolongation or taking other QTc-prolonging drugs. High doses should be avoided in elderly patients and those with electrolyte abnormalities to reduce the risk of cardiac arrhythmias.